Series A · Biotech

TwoStep Therapeutics raises $62.5m Series A for TS-104 and its cancer pipeline

Its targeting peptide binds five integrins and can carry different treatment payloads.

TwoStep Therapeutics raised $62.5 million in Series A financing, bringing cumulative funding to $71.2 million. Recorded backers include Insight Partners, Medical Excellence Capital, NFX, M Ventures, Pfizer Ventures, 2048 Ventures and Stanford University.

The company plans to advance lead peptide-drug conjugate TS-104 into Phase 1 oncology development, advance its radioligand programme and expand the peptide-conjugate pipeline.

Its polyspecific integrin-binding peptide recognises five tumour-associated integrins and can carry different treatment payloads. TS-104 links it to MMAE; the platform also supports radioligand approaches.

Use of funds

Advance lead peptide-drug conjugate TS-104 through Phase 1 oncology development

Advance radioligand program

Expand peptide-conjugate pipeline

Funding history

Series A · This round$62.5M

Sources

  1. TwoStep Therapeutics Raises $62.5M in Fundingfinsmes.com · Sep 9, 2026
  2. twosteptx.com
  3. twosteptx.com